Cyclobarbital

Cyclobarbital, also known as cyclobarbitol or cyclobarbitone, is a drug that is a barbiturate derivative.[1] It is primarily available in fixed-dose combination with diazepam under the brand name Reladorm (100 mg cyclobarbital + 10 mg diazepam) and is used to treat insomnia in Russia.[2]

Cyclobarbital

Clinical data
AHFS/Drugs.com	International Drug Names
Routes of administration	Oral (tablets)
ATC code	N05CA10 (WHO)
Legal status
Legal status	CA: Schedule IV DE: Anlage II (Authorized trade only, not prescriptible)
Pharmacokinetic data
Metabolism	Hepatic
Excretion	Renal
Identifiers
IUPAC name 5-(1-cyclohexenyl)-5-ethyl-1,3-diazinane-2,4,6-trione
CAS Number	143-76-0^N
PubChem CID	5838
ChemSpider	5632^Y
UNII	0M8A98AD9H
KEGG	D07323^N
ChEMBL	ChEMBL268164^Y
CompTox Dashboard (EPA)	DTXSID9022865
ECHA InfoCard	100.000.127
Chemical and physical data
Formula	C12H16N2O3
Molar mass	236.271 g·mol^−1
3D model (JSmol)	Interactive image
SMILES O=C1NC(=O)NC(=O)C1(/C2=C/CCCC2)CC
InChI InChI=1S/C12H16N2O3/c1-2-12(8-6-4-3-5-7-8)9(15)13-11(17)14-10(12)16/h6H,2-5,7H2,1H3,(H2,13,14,15,16,17)^Y Key:WTYGAUXICFETTC-UHFFFAOYSA-N^Y
^NY (what is this?)  (verify)

References

1. Breimer DD, Winten MA (March 1976). "Pharmacokinetics and relative bioavailability of cyclobarbital calcium in man after oral administration". European Journal of Clinical Pharmacology. 09 (5–6): 443–50. doi:10.1007/bf00606563. PMID 989475.
2. "Russian State Register of Medicines. Registration Certificate: Reladorm (diazepam + cyclobarbital). Revised 02 Sep 2013" (in Russian). Retrieved 6 March 2016.