Bromazine
Bromazine (trade names Ambodryl,[1] Ambrodil and others), also known as bromodiphenhydramine, is an antihistamine and anticholinergic.[2] It is a brominated form of diphenhydramine.
Not to be confused with Promazine.
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MedlinePlus | a682065 |
Routes of administration | Oral |
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Bioavailability | High |
Protein binding | 96% |
Metabolism | Mostly hepatic (CYP-mediated), also renal |
Elimination half-life | 1 to 4 hours |
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ECHA InfoCard | 100.003.854 |
Chemical and physical data | |
Formula | C17H20BrNO |
Molar mass | 334.257 g·mol−1 |
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References
- Baker CE (1974). Physicians' Desk Reference (28 ed.). Oradell, NJ 07649: Medical Economics Company. pp. 1076, 1081.CS1 maint: location (link)
- Maclaren WR, Bruff WC, Eisenberg BC, Weiner H, Martin WH (1955). "A clinical comparison of carbinoxamine maleate, tripelennamine hydrochloride, and bromodiphenhydramine hydrochloride in treating allergic symptoms". Annals of Allergy. 13 (3): 307–12. PMID 14377226.
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See also: Receptor/signaling modulators • Monoamine metabolism modulators • Monoamine reuptake inhibitors |
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